Inhibitors for distinction of three types of human glutathione transferase
- 25 February 1985
- journal article
- Published by Wiley in FEBS Letters
- Vol. 181 (2), 249-252
- https://doi.org/10.1016/0014-5793(85)80269-6
Abstract
A set of inhibitors that are useful for distinction of three types of human cytosolic glutathione transferase is presented. The near-neutral transferase is inhibited most effectively by Cibacron blue (itI50 = 0.05 μM), the acidic transferase by Cibacron blue (itI50 = 0.5 μM), and the basic transferase by tributyltin acetate (itI50 = 0.1 μM). The use of any of these two compounds makes possible differentiation between all three types of human transferase.Keywords
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