Use of Dibutyl[14C]formamide as a Formylating Reagent in the Vilsmeier–Haack Reaction and Synthesis of a 14C‐Labeled Novel Phosphodiesterase‐4 (PDE‐4) Inhibitor
- 18 May 2005
- journal article
- research article
- Published by Wiley in Helvetica Chimica Acta
- Vol. 88 (5), 1040-1047
- https://doi.org/10.1002/hlca.200590075
Abstract
No abstract availableKeywords
This publication has 10 references indexed in Scilit:
- Practical synthesis of a highly functionalized thiazole ketoneTetrahedron, 2003
- Optimization of a Tertiary Alcohol Series of Phosphodiesterase-4 (PDE4) Inhibitors: Structure−Activity Relationship Related to PDE4 Inhibition and Human Ether-a-go-go Related Gene Potassium Channel Binding AffinityJournal of Medicinal Chemistry, 2003
- Substituted 2-Pyridinemethanol derivatives as potent and selective phosphodiesterase-4 inhibitorsBioorganic & Medicinal Chemistry Letters, 2003
- Substituted aminopyridines as potent and selective phosphodiesterase-4 inhibitorsBioorganic & Medicinal Chemistry Letters, 2003
- Substituted 4-(2,2-diphenylethyl)pyridine-N-oxides as phosphodiesterase-4 inhibitors: SAR study directed toward the improvement of pharmacokinetic parametersBioorganic & Medicinal Chemistry Letters, 2002
- Vilsmeier formylation and glyoxylation reactions of nucleophilic aromatic compounds using pyrophosphoryl chlorideTetrahedron, 1993
- A Convenient Preparation of Pyrophosphoryl Chloride and Its Use in Vilsmeier Formylation ReactionsSynlett, 1992
- Synthesis of 5-azacytidine-6-13C and -6-14CJournal of Medicinal Chemistry, 1977
- On the bound form of ascorbic acid. XIX. Synthesis of ascorbigen-(14C)Collection of Czechoslovak Chemical Communications, 1963
- Notes. Synthesis of C14 Labelled Dimethylformamide and 3-(2-Amino-butyl-1-C14)indole Acetic Acid SaltThe Journal of Organic Chemistry, 1961