Affinity profiles of morphine, codeine, dihydrocodeine and their glucuronides at opioid receptor subtypes
- 1 January 1995
- journal article
- Published by Elsevier in Life Sciences
- Vol. 56 (10), 793-799
- https://doi.org/10.1016/0024-3205(95)00010-4
Abstract
No abstract availableKeywords
This publication has 16 references indexed in Scilit:
- The analgesic activity of morphine‐6‐glucuronide.British Journal of Clinical Pharmacology, 1992
- Morphine 6-glucuronide and morphine 3-glucuronide as molecular chameleons with unexpected lipophilicityJournal of Medicinal Chemistry, 1991
- DISPOSITION OF MORPHINE-6-GLUCURONIDE AND MORPHINE IN HEALTHY VOLUNTEERSBritish Journal of Anaesthesia, 1991
- ANALGESIC EFFICACY AND CSF PHARMACOKINETICS OF INTRATHECAL MORPHINE-6-GLUCURONIDE: COMPARISON WITH MORPHINEBritish Journal of Anaesthesia, 1990
- The spinal antinociceptive actions of morphine metabolites morphine-6-glucuronide and normorphine in the ratBrain Research, 1989
- Morphine-6-glucuronide: Analgesic effects and receptor binding profile in ratsLife Sciences, 1988
- Morphine-6-glucuronide, a potent mu agonistLife Sciences, 1987
- Enhanced binding of morphine and nalorphine to opioid delta receptor by glucuronate and sulfate conjugations at the 6-positionLife Sciences, 1987
- Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reactionBiochemical Pharmacology, 1973
- Metabolism of Drugs. LX. The Synthesis of Codeine and Morphine GlucuronidesCHEMICAL & PHARMACEUTICAL BULLETIN, 1968