Docetaxel (taxotere) derivatives: novel NbCl3-based stereoselective approach to 2′-methyldocetaxel
- 1 January 1995
- journal article
- research article
- Published by Royal Society of Chemistry (RSC) in Journal of the Chemical Society, Perkin Transactions 1
- No. 14,p. 1811-1815
- https://doi.org/10.1039/p19950001811
Abstract
The C-2 methylated 2S,3R and 2R,3S side chains of docetaxel have been enantioselectively prepared and esterified with protected 10-deacetylbaccatin III to provide novel analogues of docetaxel.Keywords
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