Probing the P3′ pocket of stromelysin with piperazic acid analogs
- 21 December 1995
- journal article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 5 (24), 3053-3056
- https://doi.org/10.1016/0960-894x(95)00536-1
Abstract
No abstract availableKeywords
This publication has 12 references indexed in Scilit:
- Inhibition of matrix metalloproteinases by N-carboxyalkyl peptides containing extended alkyl residues At P1'Bioorganic & Medicinal Chemistry Letters, 1995
- Inhibition of Human Stromelysin by Peptides Based on the N-Terminal Domain of Tissue Inhibitor of Metalloproteinases-1Biochemical and Biophysical Research Communications, 1994
- Inhibition of stromelysin-1 (MMP-3) by peptidyl phosphinic acidsBioorganic & Medicinal Chemistry Letters, 1994
- Inhibition of Matrix Metalloproteinases by Peptidyl Hydroxamic AcidsBiochemical and Biophysical Research Communications, 1994
- Matlystatins, new inhibitors of type IV collagenases from Actinomadura atramentaria. IV. Synthesis and structure-activity relationships of matlystatin b and its stereoisomers.The Journal of Antibiotics, 1994
- Azinothricin synthetic studies. 1. Efficient asymmetric synthesis of (3R)- and (3S)-piperazic acidsTetrahedron Letters, 1992
- Cloning of the genes for human stromelysin and stromelysin 2: differential expression in rheumatoid synovial fibroblastsBiochemistry, 1989
- Purification of the neutral proteoglycan-degrading metalloproteinase from human articular cartilage tissue and its identification as stromelysin matrix metalloproteinase-3Biochemical Journal, 1989
- Human skin fibroblast stromelysin: structure, glycosylation, substrate specificity, and differential expression in normal and tumorigenic cells.Proceedings of the National Academy of Sciences, 1987
- Asymmetric alkylation reactions of chiral imide enolates. A practical approach to the enantioselective synthesis of .alpha.-substituted carboxylic acid derivativesJournal of the American Chemical Society, 1982