Characterization of a Set of HIV-1 Protease Inhibitors Using Binding Kinetics Data from a Biosensor-Based Screen
Open Access
- 1 October 2000
- journal article
- research article
- Published by Elsevier in SLAS Discovery
- Vol. 5 (5), 353-359
- https://doi.org/10.1177/108705710000500507
Abstract
No abstract availableKeywords
This publication has 14 references indexed in Scilit:
- Kinetic Analysis of the Interaction between HIV-1 Protease and Inhibitors Using Optical Biosensor TechnologyAnalytical Biochemistry, 2000
- Design and Fast Synthesis of C-Terminal Duplicated PotentC2-Symmetric P1/P1‘-Modified HIV-1 Protease InhibitorsJournal of Medicinal Chemistry, 1999
- Screening of Compounds Interacting with HIV-1 Proteinase Using Optical Biosensor TechnologyAnalytical Biochemistry, 1998
- Design and Synthesis of New PotentC2-Symmetric HIV-1 Protease Inhibitors. Use ofl-Mannaric Acid as a Peptidomimetic ScaffoldJournal of Medicinal Chemistry, 1998
- HIV-1 Protease Inhibitors Based on Acyclic CarbohydratesThe Journal of Organic Chemistry, 1998
- Synthesis of enantiomerically pure cis and trans 2-aminocyclopentanecarboxylic acids. Use of proline replacements in potential HIV-protease inhibitorsTetrahedron, 1997
- A convenient synthesis of 1-(S)-[1′-(S)-(t-butyloxycarbonylamino)-2′-phenylethyl]oxirane. A useful building block in the synthesis of HIV protease inhibitorsTetrahedron Letters, 1997
- Cyclic HIV-1 Protease Inhibitors Derived from Mannitol: Synthesis, Inhibitory Potencies, and Computational Predictions of Binding AffinitiesJournal of Medicinal Chemistry, 1997
- Synthesis ofC2Symmetric Potential Inhibitors of HIV-1 Protease From D-MannitolJournal of Carbohydrate Chemistry, 1996
- Biospecific interaction analysis using surface plasmon resonance detection applied to kinetic, binding site and concentration analysisJournal of Chromatography A, 1992