Synthesis and evaluation of benzophenone-based photoaffinity labeling analogs of prenyl pyrophosphates containing stable amide linkages
- 19 August 1997
- journal article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 7 (16), 2125-2130
- https://doi.org/10.1016/s0960-894x(97)00373-9
Abstract
No abstract availableKeywords
This publication has 19 references indexed in Scilit:
- Analogs of farnesyl pyrophosphate incorporating internal benzoylbenzoate esters: Synthesis, inhibition kinetics and photoinactivation of yeast protein farnesyltransferaseTetrahedron Letters, 1996
- PROTEIN PRENYLATION: Molecular Mechanisms and Functional ConsequencesAnnual Review of Biochemistry, 1996
- Photoactive Analogs of Farnesyl Pyrophosphate Containing Benzoylbenzoate Esters: Synthesis and Application to Photoaffinity Labeling of Yeast Protein FarnesyltransferaseThe Journal of Organic Chemistry, 1996
- Farnesyl transferase inhibitors: the successes and surprises of a new class of potential cancer chemotherapeuticsChemistry & Biology, 1995
- Chemical reagents in photoaffinity labelingTetrahedron, 1995
- Photoreactive Analogues of Prenyl Diphosphates as Inhibitors and Probes of Human Protein Farnesyltransferase and Geranylgeranyltransferase Type IPublished by Elsevier ,1995
- Mammalian Protein Geranylgeranyltransferase-I: Substrate Specificity, Kinetic Mechanism, Metal Requirements, and Affinity LabelingBiochemistry, 1995
- Farnesyltransferase inhibitors: Ras research yields a potential cancer therapeuticCell, 1994
- Characterization of recombinant human farnesyl-protein transferase: Cloning, expression, farnesyl diphosphate binding, and functional homology with yeast prenyl-protein transferasesBiochemistry, 1993
- Inhibition of farnesyl transferases from malignant and non-malignant cultured human lymphocytes by prenyl substrate analoguesBiochemical and Biophysical Research Communications, 1991