8-Aminocyclazocine analogues: synthesis and structure–activity relationships
- 17 January 2000
- journal article
- research article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 10 (2), 183-187
- https://doi.org/10.1016/s0960-894x(99)00670-8
Abstract
No abstract availableKeywords
This publication has 16 references indexed in Scilit:
- Transition Metal Catalyzed Synthesis of Arylamines and Aryl Ethers from Aryl Halides and Triflates: Scope and MechanismAngewandte Chemie International Edition, 1998
- Palladium-Catalyzed Amination of Aryl Triflates and Importance of Triflate Addition RateThe Journal of Organic Chemistry, 1997
- Palladium-Catalyzed Amination of Aryl TriflatesThe Journal of Organic Chemistry, 1997
- Synthesis and .sigma. Binding Properties of 2'-Substituted 5,9.alpha.-Dimethyl-6,7-benzomorphansJournal of Medicinal Chemistry, 1995
- 14.alpha.,14'.beta.-[Dithiobis[(2-oxo-2,1-ethanediyl)imino]]bis(7,8-dihydromorphinone) and 14.alpha.,14'.beta.-[Dithiobis[(2-oxo-2,1-ethanediyl)imino]]bis-7,8-dihydro-N-(cyclopropyl- methyl)normorphinone: Chemistry and Opioid Binding PropertiesJournal of Medicinal Chemistry, 1994
- Synthesis and evaluation of 3-substituted 17-methylmorphinan analogs as potential anticonvulsant agentsJournal of Medicinal Chemistry, 1992
- Affinity of the enantiomers of α- and β-cyclazocine for binding to the phencyclidine and μ opioid receptorsLife Sciences, 1990
- Synthesis and evaluation of optically pure [3H]‐(+)‐pentazocine, a highly potent and selective radioligand for σ receptorsFEBS Letters, 1989
- Synthesis and pharmacology of 8-amino-3-(cyclopropylmethyl)-1,2,3,4,5,6-hexahydro-cis-6,11-dimethyl-2,6-methano-3-benzazocine and related compoundsJournal of Medicinal Chemistry, 1980
- Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reactionBiochemical Pharmacology, 1973