Potent inhibition of thrombin by the newly synthesized arginine derivative No. 805. The importance of stereo-structure of its hydrophobic carboxamide portion
- 1 July 1981
- journal article
- research article
- Published by Elsevier in Biochemical and Biophysical Research Communications
- Vol. 101 (2), 440-446
- https://doi.org/10.1016/0006-291x(81)91279-1
Abstract
No abstract availableKeywords
This publication has 10 references indexed in Scilit:
- Thrombin inhibitors. 3. Carboxyl-containing amide derivatives of N.alpha.-substituted L-arginineJournal of Medicinal Chemistry, 1980
- Thrombin inhibitors. 1. Ester derivatives of N.alpha.-(arylsulfonyl)-L-arginineJournal of Medicinal Chemistry, 1980
- Thrombin inhibitors. 2. Amide derivatives of N.alpha.-substituted L-arginineJournal of Medicinal Chemistry, 1980
- Kinetic Studies on the Selectivity of a Synthetic Thrombin-Inhibitor Using Synthetic Peptide SubstratesThrombosis and Haemostasis, 1979
- Diarylamidine derivatives with one or both of the aryl moieties consisting of an indole or indole-like ring. Inhibitors of arginine-specific esteroproteasesJournal of Medicinal Chemistry, 1978
- Synthetic inhibitors of serine proteinases XVI. Influence of 3- and 4-amidinobenzyl derivatives on the formation and action of thrombinThrombosis Research, 1978
- Aromatic esters which inhibit plasmin or thrombin by formation of relatively stable acyl enzymesJournal of Medicinal Chemistry, 1973
- Differential specificities of thrombin, plasmin and trypsin with regard to synthetic and natural substrates and inhibitorsBiochimica et Biophysica Acta (BBA) - Enzymology, 1972
- Rapid method for the purification of bovine thrombin and the inhibition of the purified enzyme with phenylmethylsulfonyl fluorideBiochemistry, 1971
- 422. Experiments towards the synthesis of corrins. Part I. The preparation and reactions of some Δ1-pyrrolines. A novel proline synthesisJournal of the Chemical Society, 1959