Synthesis of RPR 100893, prototype of a new series of potent and selective non peptide NK1 antagonists : the triarylperhydroisoindolols.
- 10 March 1994
- journal article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 4 (5), 673-676
- https://doi.org/10.1016/s0960-894x(01)80178-5
Abstract
No abstract availableKeywords
This publication has 18 references indexed in Scilit:
- Antinociceptive properties and inhibition of neurogenic inflammation with potent SP antagonists belonging to perhydroisoindolonesRegulatory Peptides, 1993
- Inhibition of neurogenic inflammation in the meninges by a non-peptide NK1 receptor antagonist, RP 67580European Journal of Pharmacology, 1993
- Synthesis of RP-67,580, a new potent nonpeptide substance P antagonistBioorganic & Medicinal Chemistry Letters, 1992
- The discovery of (2S,3S)-cis-2-(diphenylmethyl)-N-[(2-methoxyphenyl)methyl]-1-azabicyclo[2.2.2]octan-3-amine as a novel, nonpeptide substance P antagonistJournal of Medicinal Chemistry, 1992
- Tachykinin receptor types: Classification and membrane signalling mechanismsNeurochemistry International, 1991
- Modulation of neurogenic inflammation: novel approaches to inflammatory diseaseTrends in Pharmacological Sciences, 1990
- TachykininsAnnual Review of Neuroscience, 1988
- Does substance P act as a pain transmitter?Trends in Pharmacological Sciences, 1987
- cDNA eloping of bovine substance-K receptor through oocyte expression systemNature, 1987
- Substance P as a Transmitter CandidateAnnual Review of Neuroscience, 1980