Synthesis of [d-ALA2, 4′-125I-PHE3, GLU4] deltorphin and characterization of its δ opioid receptor binding properties
- 31 December 1992
- journal article
- Published by Elsevier in Life Sciences
- Vol. 51 (20), PL189-PL193
- https://doi.org/10.1016/0024-3205(92)90628-3
Abstract
No abstract availableKeywords
This publication has 9 references indexed in Scilit:
- Synthesis and binding characteristics of the highly delta-specific new tritiated opioid peptide, [3H] deltorphin IILife Sciences, 1992
- Topographical requirements for delta opioid ligands: Presence of a carboxyl group in position 4 is not critical for deltorphin high delta receptor affinity and analgesic activityBiochemical and Biophysical Research Communications, 1991
- A simple general method for (radio)iodination of a phenylalanine residue in peptides: preparation of [cyclic][D-Pen2,4'-125I-Phe4,D-Pen5]enkephalin, a peptide with extraordinary selectivity for .delta.-opioid receptorsThe Journal of Organic Chemistry, 1991
- Evidence for two subtypes of δ opioid receptors in rat brainEuropean Journal of Pharmacology, 1991
- [Cyclic] [D-Pen2,D-Pen5]enkephalin analogs with increased affinity and selectivity for .delta.-opioid receptorsJournal of Medicinal Chemistry, 1990
- Deltorphin, a novel amphibian skin peptide with high selectivity and affinity for δ opioid receptorsEuropean Journal of Pharmacology, 1989
- Dermorphin Gene Sequence Peptide with High Affinity and Selectivity for δ-Opioid ReceptorsPublished by Elsevier ,1989
- The use of [3H]‐[d‐Pen2,d‐Pen5]enkephalin as a highly selective ligand for the δ‐binding siteBritish Journal of Pharmacology, 1985
- Selectivities of opioid peptide analogues as agonists and antagonists at the δ‐receptorBritish Journal of Pharmacology, 1984