A versatile synthesis of a β-turn peptidomimetic scaffold: An approach towards a designed model antagonist of the tachykinin NK-2 receptor
- 9 July 1996
- journal article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 6 (13), 1567-1572
- https://doi.org/10.1016/s0960-894x(96)00275-2
Abstract
No abstract availableKeywords
This publication has 43 references indexed in Scilit:
- Electrochemical Cyclization of Dipeptides To Form Novel Bicyclic, Reverse-Turn Peptidomimetics. 2. Synthesis and Conformational Analysis of 6,5-Bicyclic SystemsThe Journal of Organic Chemistry, 1996
- Stereoselective Approaches to Bioactive Carbohydrates and Alkaloids-With a Focus on Recent Syntheses Drawing from the Chiral PoolChemical Reviews, 1995
- Furan-, Pyrrole-, and Thiophene-Based Siloxydienes for Syntheses of Densely Functionalized Homochiral CompoundsSynthesis, 1995
- A facile synthesis of the novel Neurokinin A antagonist SR 48968Bioorganic & Medicinal Chemistry Letters, 1993
- Cyclic peptides as selective tachykinin antagonistsJournal of Medicinal Chemistry, 1993
- A new class of high affinity ligands for the neurokinin A NK2 receptor: .psi.(CH2NR) reduced peptide bond analogs of neurokinin A4-10Journal of Medicinal Chemistry, 1992
- Conformation of a neurokinin antagonist in solutionInternational Journal of Peptide and Protein Research, 1992
- Neurokinin A (NK2) receptor revisited with SR 48968, a potent non-peptide antagonistBiochemical and Biophysical Research Communications, 1992
- Are the proposed substance P receptor sub-types, substance P receptors?Life Sciences, 1984
- The tachykinin peptide familyTrends in Neurosciences, 1981