Solubilization of Thiazolobenzimidazole Using a Combination of pH Adjustment and Complexation with 2-Hydroxypropyl-β-Cyclodextrin

Abstract
The thiazolobenzimidazole l-(2,6-difluorophenyl)-lH,3H-thiazolo[3,4- a]benzimidazole, TBI, is an experimental drug for the treatment of AIDS which exhibits a low water solubility (11 µg/mL) and is...