UNEXPECTED ANTAGONISM IN THE RAT VAS DEFERENS BY BENZOMORPHANS WHICH ARE AGONISTS IN OTHER PHARMACOLOGICAL TESTS
Open Access
- 1 January 1981
- journal article
- Published by Wiley in British Journal of Pharmacology
- Vol. 72 (1), 13-15
- https://doi.org/10.1111/j.1476-5381.1981.tb09098.x
Abstract
The benzomorphans, ethylketazocine, bremazocine and MR 2034 are pure agonists in the guinea-pig ileum and mouse vas deferens but are competitive antagonists without agonist activity in the rat vas deferens.Keywords
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