Diastereomeric Fluoroolefins as Peptide Bond Mimics Prepared by Asymmetric Reductive Amination of α‐Fluoroenones
- 5 February 2007
- journal article
- research article
- Published by Wiley in Angewandte Chemie International Edition
- Vol. 46 (8), 1290-1292
- https://doi.org/10.1002/anie.200604246
Abstract
No abstract availableKeywords
This publication has 37 references indexed in Scilit:
- Fluoroolefins as Peptide Mimetics: A Computational Study of Structure, Charge Distribution, Hydration, and Hydrogen BondingThe Journal of Physical Chemistry A, 2006
- Synthesis and biological evaluation of γ-fluoro-β,γ-unsaturated acidsJournal of Fluorine Chemistry, 2006
- Fluoro-Olefins as Peptidomimetic Inhibitors of Dipeptidyl PeptidasesJournal of Medicinal Chemistry, 2004
- Toward (Z)-selective Horner–Wadsworth–Emmons reaction of aldehydes with 2-fluoro-2-diethylphosphonoacetic acidTetrahedron Letters, 2002
- Formation of Enantiomerically Pure 1-Fluorovinyl and 1-Fluoromethyl SulfoxidesEuropean Journal of Organic Chemistry, 2001
- Fluoroalkenes as Peptide Isosteres: Ground State Analog Inhibitors of ThermolysinThe Journal of Organic Chemistry, 1995
- Fluoroolefin peptide isosteres - tools for controlling peptide conformationsTetrahedron Letters, 1994
- Stereospecific method to (E) and (Z) terminal fluoroolefins and its application to the synthesis of 2'-deoxy-2'-fluoromethylenenucleosides as potential inhibitors of ribonucleoside diphosphate reductaseJournal of the American Chemical Society, 1991
- Fluoroolefin dipeptide isosteres -II. : Enantioselectlve synthesis of both antipodes of the phe-gly dlpeptide mimicTetrahedron Letters, 1990
- Fluoroolefin dipeptide isosteres — I.Tetrahedron Letters, 1990