The estradiol pharmacophore: Ligand structure-estrogen receptor binding affinity relationships and a model for the receptor binding site
- 1 March 1997
- Vol. 62 (3), 268-303
- https://doi.org/10.1016/s0039-128x(96)00242-5
Abstract
No abstract availableKeywords
This publication has 202 references indexed in Scilit:
- Estrogen and androgen receptor binding affinity of 10β-chloro-estrenen derivativesThe Journal of Steroid Biochemistry and Molecular Biology, 1988
- Differential inhibition of estrogen and antiestrogen binding to the estrogen receptor by diethylpyrocarbonateThe Journal of Steroid Biochemistry and Molecular Biology, 1988
- Interaction of the antioestrogen ICI 164,384 with the oestrogen receptorJournal of Steroid Biochemistry, 1988
- Shielding effects at 17α-substituted estrogens. A tentative explanation for the low biological activity of 17α-ethyl-estradiol based on I.R. and NMR spectroscopic studiesThe Journal of Steroid Biochemistry and Molecular Biology, 1985
- Steroid binding to the cytosolic estrogen receptor from rat uterus. influence of the orientation of substituents in the 17-position of the 8β- and 8α-seriesThe Journal of Steroid Biochemistry and Molecular Biology, 1985
- Substituted derivatives of a-nor-5α-androstane and a-nor-5α-estrane—structure and affinity for hormonal receptorsThe Journal of Steroid Biochemistry and Molecular Biology, 1983
- Steroid structure and function—IX. Molecular conformation and receptor binding of isomeric analogs of d-Homo-EstradiolThe Journal of Steroid Biochemistry and Molecular Biology, 1980
- The androgen receptor binding site: A conformational study of steroids in relation with their affinity—I. Interaction with the D-ringThe Journal of Steroid Biochemistry and Molecular Biology, 1980
- A series of optical, structural and isomeric analogs of estradiol: A comparative study of the biological activity and affinity to cytosol receptor of rabbit uterusThe Journal of Steroid Biochemistry and Molecular Biology, 1975
- The specificity of the estrogen receptor of human uterusJournal of Steroid Biochemistry, 1973