Regiospecific Synthesis of Certain 1,2,3,4-Tetrasubstituted Benzenes in One Step via a Benzene Cyclization
- 1 January 1989
- journal article
- research article
- Published by Taylor & Francis in Synthetic Communications
- Vol. 19 (1-2), 233-237
- https://doi.org/10.1080/00397918908050974
Abstract
Tetrasubstituted benzenes of type 3 are obtained regiospecifically in a single step by the treatment of 1-fluoro-4-methoxy-5-carbo-tert-butoxy aniline with tert-butyllithium followed by reaction with an electrophile.Keywords
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