Rational design of potent carboxylic acid based bisubstrate inhibitors of ras farnesyl protein transferase
- 8 September 1994
- journal article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 4 (17), 2107-2112
- https://doi.org/10.1016/s0960-894x(01)80111-6
Abstract
No abstract availableKeywords
This publication has 8 references indexed in Scilit:
- Benzodiazepine Peptidomimetics: Potent Inhibitors of Ras Farnesylation In Animal CellsScience, 1993
- Selective Inhibition of ras -Dependent Transformation by a Farnesyltransferase InhibitorScience, 1993
- Tetrapeptide inhibitors of protein farnesyltransferase: amino-terminal substitution in phenylalanine-containing tetrapeptides restores farnesylation.Proceedings of the National Academy of Sciences, 1992
- Steady-state kinetic mechanism of ras farnesyl:protein transferaseBiochemistry, 1992
- Identification and preliminary characterization of protein-cysteine farnesyltransferase.Proceedings of the National Academy of Sciences, 1990
- Syntheses and reactions of silyl carbamates. 1. Chemoselective transformation of amino protecting groups via tert-butyldimethylsilyl carbamatesThe Journal of Organic Chemistry, 1990
- Stereospecific amino acid synthesis; preparation of the γ-anion derived from glutamic acidJournal of the Chemical Society, Chemical Communications, 1988
- ras GENESAnnual Review of Biochemistry, 1987