Lewis acid promoted regio- and stereoselective hetero nucleophilic addition to a piperidinyl aziridine. Synthesis of trans 3-amino-4-substituted piperidines
- 9 June 2002
- journal article
- research article
- Published by Elsevier in Tetrahedron Letters
- Vol. 43 (30), 5315-5318
- https://doi.org/10.1016/s0040-4039(02)01024-9
Abstract
No abstract availableThis publication has 17 references indexed in Scilit:
- Regio- and stereo-controlled copper organometallic addition to a piperidinyl aziridine: synthesis of trans 3-amino-4-alkyl-piperidinesTetrahedron Letters, 2002
- Effective Ring-Opening Reaction of Aziridines with Trimethylsilyl Compounds: A Facile Access to β-Amino Acids and 1,2-Diamine DerivativesThe Journal of Organic Chemistry, 2000
- Novel Synthesis of 4-Carboxymethyl 5-Alkyl/Aryl Oxazolidin-2-ones by Rearrangement of 2-Carboxymethyl 3-Alkyl/ArylN-tert-Butoxycarbonyl AziridinesOrganic Letters, 1999
- General Syntheses of Optically Active α-Trifluoromethylated Amines via Ring-Opening Reactions of N-Benzyl-2-trifluoromethylaziridineThe Journal of Organic Chemistry, 1999
- Conformationally Constrained 1,3-Diamino Ketones: A Series of Potent Inhibitors of the Cysteine Protease Cathepsin KJournal of Medicinal Chemistry, 1998
- 2,3-Aziridino-2,3-dideoxy-d-ribono-γ-lactone 5-Phosphonate: Stereocontrolled Synthesis from d-Lyxose and Unusual Aziridine Ring OpeningThe Journal of Organic Chemistry, 1997
- An efficient stereoselective synthesis of the amino sugar component (E ring) of calicheamicin γ1ITetrahedron: Asymmetry, 1996
- Synthetic Studies towards A trans-3,4-Diamine Derivative of Piperidine Mimicking BuspironeHETEROCYCLES, 1994
- trans-3,4-Diaminopiperidines. Azacyclohexane congeners of .kappa. agonist U-50488The Journal of Organic Chemistry, 1991
- Synthesis of side-chain monofluorinated amphetaminesJournal of Fluorine Chemistry, 1980