Palladium-catalyzed tandem C,N-arylation of immobilized enamine for solid phase indole synthesisElectronic supplementary information (ESI) available: experimental procedures. See http://www.rsc.org/suppdata/p1/b2/b206378f/

Abstract

Intramolecular palladium-catalyzed N-arylation of immobilized dehydrohalophenylalaninate was found to proceed smoothly to form indolecarboxylates. The method was successfully combined with the Heck reaction to perform one pot indole synthesis via palladium-catalyzed tandem C,N-arylation reactions.