A Synthesis of RGD Model Cyclic Peptide by Palladium-Catalyzed Carbonylative Macrolactamization
- 31 January 2008
- journal article
- Published by American Chemical Society (ACS) in Organic Letters
- Vol. 10 (5), 817-819
- https://doi.org/10.1021/ol702965r
Abstract
Cyclic peptidic RGD models were efficiently synthesized by Pd(P(t-Bu)3)2-catalyzed carbonylative macrolactamization in the presence of 4 Å molecular sieves under 10 atm of carbon monoxide.Keywords
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