Organocatalytic Conjugate Addition of Malonates to α,β‐Unsaturated Aldehydes: Asymmetric Formal Synthesis of (−)‐Paroxetine, Chiral Lactams, and Lactones
Top Cited Papers
- 16 June 2006
- journal article
- research article
- Published by Wiley in Angewandte Chemie International Edition
- Vol. 45 (26), 4305-4309
- https://doi.org/10.1002/anie.200601025
Abstract
No abstract availableKeywords
This publication has 59 references indexed in Scilit:
- Taking inventory: antibacterial agents currently at or beyond Phase 1Current Opinion in Microbiology, 2004
- A Convenient Synthesis of (−)‐ParoxetineEuropean Journal of Organic Chemistry, 2004
- Structural differences between paroxetine and femoxetine responsible for differential inhibition of Staphylococcus aureus efflux pumpsBioorganic & Medicinal Chemistry Letters, 2004
- Effect of Microwaves in the Chiral Switching Asymmetric Michael ReactionMolecules, 2003
- Synthesis of Enantiopuretrans-3,4-Disubstituted Piperidines. An Enantiodivergent Synthesis of (+)- and (−)-ParoxetineThe Journal of Organic Chemistry, 2000
- Reductive Amination of Aldehydes and Ketones with Sodium Triacetoxyborohydride. Studies on Direct and Indirect Reductive Amination Procedures1The Journal of Organic Chemistry, 1996
- Overview Central & Peripheral Nervous System: Recent developments in serotonin reuptake inhibitorsExpert Opinion on Therapeutic Patents, 1994
- Synthesis and use of 3-amino-4-phenyl-2-piperidones and 4-amino-2-benzazepin-3-ones as conformationally restricted phenylalanine isosteres in renin inhibitorsJournal of Medicinal Chemistry, 1992
- .beta.-Substituted .beta.-phenylpropionyl chymotrypsins. Structural and stereochemical features in stable acyl enzymesJournal of Medicinal Chemistry, 1991
- The Michael addition of dimethyl malonate to α,β-unsaturated aldehydes catalysed by proline lithium saltJournal of the Chemical Society, Chemical Communications, 1991